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First in class (S,E)-11-[2-(arylmethylene)hydrazono]-PBD analogs as selective CB2 modulators targeting neurodegenerative disorders

  • David Mingle
  • , Meirambek Ospanov
  • , Mohamed O. Radwan
  • , Nicole Ashpole
  • , Masami Otsuka
  • , Samir A. Ross
  • , Larry A. Walker
  • , Abbas G. Shilabin
  • , Mohamed A. Ibrahim
  • East Tennessee State University
  • University of Mississippi School of Pharmacy
  • Kumamoto University
  • Science Farm Ltd.
  • National Research Centre

Research output: Contribution to journalArticlepeer-review

Original languageEnglish
Pages (from-to)98-108
Number of pages11
JournalMedicinal Chemistry Research
Volume30
Issue number1
DOIs
StatePublished - Jan 2021

ASJC Scopus Subject Areas

  • General Pharmacology, Toxicology and Pharmaceutics
  • Organic Chemistry

Keywords

  • Cannabinoid receptors CB1/CB2
  • Central nervous system (CNS)
  • Neurodegenerative diseases
  • Neuroinflammation
  • Pyrrolobenzodiazepines

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